99% Tianeptine sodium gishiri CAS 30123-17-2
Ƙayyadaddun bayanai
ITEM | STANDARD | SAKAMAKO |
Bayyanar | Fari zuwa foda mai rawaya | Farar crystalline foda |
Solubility | Soluble A cikin ruwa da methanol da dichloromethane | Ya dace |
Ganewa | Ta IR, Don dacewa da daidaitattun aiki | Ya dace |
(2) Yana ba da amsawar sodium | Ya dace | |
Kayayyakin A | ≤0.1% | Ba a gano ba |
Abubuwan da ke da alaƙa | Duk wani mafi girman ƙazanta ≤0.1% | 0.060% |
Jimlar ƙazanta ≤0.4% | 0.36% | |
Residual Solvents (GC) | Acetidin ≤ 0.5% | ND |
Dichloromethane ≤ 0.06% | ND | |
Methanol ≤ 0.3% | ND | |
Acetone 0.5% | 0.29% | |
Acetonitrile ≤0.041% | 0.022% | |
Ethanol ≤0.5% | ND | |
N, N-dimethylformamide≤0.088% | ND | |
Ruwa | ≤ 5.0% | 3.8% |
Assay (HPLC) | 99.0% -101.0% (A kan anhydrousbasis) | 99.70% |
Aikace-aikace
Tianeptine sodiumgishirishi ne tricyclic antidepressant.Tsarinsa na maganin damuwa ya bambanta da na gargajiya na tricyclic antidepressants.Zai iya ƙara sake ɗaukan 5-HT a cikin ɓangarorin synaptic.Sakamakon HT neuronal conduction.Babu kusanci ga choline ko masu karɓar adrenergic.Amfanin maganin damuwa yana kama da na tricyclics, amma haƙuri ya fi na tricyclics.Don maganin rashin tausayi, matsakaici ko matsananciyar damuwa, neurogenic da damuwa mai amsawa, damuwa da damuwa tare da jiki, musamman rashin jin daɗi na gastrointestinal, da damuwa da damuwa a cikin marasa lafiya masu shan barasa a lokacin janyewa.